WebSep 6, 2024 · (A) Voltage family current trace of WT Eag1, Eag1TM, and the Eag1/hErg chimera with the voltage-pulse protocol shown above. (B) Normalized tail current vs. depolarization voltage plot for WT Eag1 (black square, n = 6), Eag1TM (green circle, n = 4), and the Eag1/hErg chimera (red triangle, n = 4) with V 0.5 values (mean ± sd).Eag1TM … WebEther-à-go-go-1 (Eag1) is an ion channel that plays important roles in tumour proliferation, malignant transformation, invasion, metastasis, recurrence, and prognosis. Therefore, identifying potent and specific Eag1 channel inhibitors is crucial. In this study, we identified the first natural inhibitor of Eag1, the traditional Chinese medicine ...
Regulation of Eag1 gating by its intracellular domains eLife
WebProduct Source An E. coli strain that carries the cloned and modified EagI gene from Enterobacter agglomerans (R. Morgan) This product is related to the following categories: Restriction Endonucleases C G, High-Fidelity (HF®) Restriction Endonucleases Products, Time-Saver Qualified Restriction Enzymes Products WebEag1 (ether-à-go-go-1), a member of the voltage-dependent potassium channel family, is expressed mainly in the brain, and at low levels in placenta, testis, and adrenal gland, and only transiently in myoblasts. Recently, several studies have suggested that Eag1 is selectively expressed in various tu … how to reset a suunto core watch
Overexpression of Eag1 potassium channels in clinical …
WebMar 13, 2008 · Abstract. Emerging evidence indicates that ion channels act in a variety of physiologic and pathologic processes beyond electronic signal transmission, including in … WebSep 12, 2012 · Background Calcitriol antiproliferative effects include inhibition of the oncogenic ether-à-go-go-1 potassium channel (Eag1) expression, which is necessary for cell cycle progression and tumorigenesis. Astemizole, a new promising antineoplastic drug, targets Eag1 by blocking ion currents. Herein, we characterized the interaction between … WebSep 24, 2024 · By contrast, Eag1 channel expression has also been demonstrated in over 70% various clinical tumours [14,15]. Eag1 is involved in cell proliferation, survival, angiogenesis, migration and invasion of cancer cells [16,17]. The expression of Eag1 is regulated by Nutlin-3 through p38 MAPK/p53 pathway [18] and/or p53-miR-34-E2F1 … north carolina not for profit